序号 | 企业代号 | 中文名 | 英文名 | CAS No. | 结构式 | 用途 |
01 | AL-5 | 2-羟基-3-甲氧基-3,3-二苯基丙酸 | 2-hydroxy-3-methoxy-3,3-diphenylpropanoic acid | 178306-51-9 | 安立生坦中间体 | |
02 | AL-6 | (S)-2-羟基-3-甲氧基-3,3-二苯基丙酸 | (S)-2-hydroxy-3-methoxy-3,3-diphenylpropanoic acid | 178306-52-9 | 安立生坦中间体 | |
03 | AMB-1 | 安立生坦 | Ambrisentan | 177036-94-1 | API | |
04 | MK-6 | 5'-甲氧基劳丹素; 6,7-二甲氧基-2-二甲基-1-(3,4,5-三甲氧基苯基)-1,2,3,4-四氢异喹啉 | 6,7-dimethoxy-2-methyl-1-(3,4,5-trimethoxybenzyl)-1,2,3,4-tetrahydroisoquinoline | 24734-71-2 | 米库氯铵中间体 | |
05 | MK-7a | (R)-N-甲基-6,7-二甲氧基-1-(3',4',5'-三甲氧基苄基)-1,2,3,4-四氢异喹啉-2,3-二苯甲酰基-L-酒石酸盐 | (R)-N-methyl-6,7-dimethoxy-1-(3',4',5'-trimethoxybenzyl)-1,2,3,4-tetrahydroisoquinolinium 2,3-dibenzoyl-L-tartarate | 米库氯铵中间体 | ||
06 | MK-8 | 2-氯化-(1R)-2-(3-羟丙基)-6,7-甲氧基-2-甲基-1-(3,4,5-三甲氧基苯基)-1,2,3,4-四氢异喹啉 | (1R)-2-(3-hydroxypropyl)-6,7-dimethoxy-2-methyl-1-(3,4,5-trimethoxybenzyl)-1,2,3,4-tetrahydroisoquinolin-2-ium chloride | 米库氯铵中间体 | ||
07 | MK-1 | 1,2,3,4-四氢-2-(3-羟丙基)-6,7-二甲氧基-2-甲基-1-(3,4,5-三甲基苄基)异喹啉氯化物(E)-4-辛烯二羧酸(2:1) | [R-[R*,R*-(E)]]-2,2'-(1,8-dioxo-4-octene-1,8-diyl)-bis(oxy-3,1-propanediyl)-bis(1,2,3,4-tetrahydro-6,7-dimethoxy-2-methyl-1-[(3,4,5-trimethoxyphenyl)-methyl]isoquinolinium) dichlorid | 106861-44-3 | API | |
08 | VON-4 | 5-(2-氟苯基)-1-(吡啶-3-基磺酰基)-3-氰基-1H-吡咯 | 5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrole-3-carbonitrile | 富马酸氟呐普拉赞中间体 | ||
09 | VON-5 | 5-(2-氟苯基)-1-(吡啶-3-基磺酰基)-1H-吡咯-3-甲醛 | 5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrole-3-carbaldehyde | 881677-11-8 | 富马酸氟呐普拉赞中间体 | |
10 | VON-1 | 富马酸氟呐普拉赞; 富马酸沃诺拉赞 | Vonoprazan Fumarate | 1260141-27-2 | API | |
11 | ATA-4 | 2-[N-(2,4,5-三甲氧基苯甲酰基)氨基]-4-乙氧基羰基-1,3-噻唑 | ethyl 2-(2,4,5-trimethoxybenzamido)thiazole-4-carboxylate | 185105-98-0 | 阿考替胺中间体 | |
12 | ATA-5 | 2-[N-(2-羟基-4,5-二甲氧基苯甲酰基)氨基]-4-乙氧基羰基-1,3-噻唑 | ethyl 2-(2-hydroxy-4,5-dimethoxybenzamido)thiazole-4-carboxylate | 阿考替胺中间体 | ||
13 | ATA-1 | 盐酸阿考替胺 | Acotiamide Hydrochloride Hydrate | 773092-05-0 | API | |
14 | ADX-2 | 2-羟基-2,2-二(噻吩-2-基)乙酸甲酯 | methyl 2-hydroxy-2,2-di(thiophen-2-yl)acetate | 阿地溴铵中间体 | ||
15 | ADX-3 | 2-羟基-2,2-二噻吩-2-基乙酸-1-单杂二环[2.2.2]辛-3(R)基酯 | (R)-quinuclidin-3-yl 2-hydroxy-2,2-di(thiophen-2-yl)acetate | 阿地溴铵中间体 | ||
16 | ADX-1 | 阿地溴铵 | Aclidinium Bromide | 320345-99-1 | API | |
17 | DT-1 | 地夸磷索钠 | Diquafosol tetrasodium | 59985-21-6 | API | |
18 | IBAN-2 | 3-(N-甲基-N-正戊胺基)丙腈 | 3-(methyl(pentyl)amino)propanenitrile | 1185103-36-9 | 伊班膦酸钠中间体 | |
19 | IBAN-3 | 3-(N-甲基正戊胺基)丙酸盐酸盐 | 3-(methyl(pentyl)amino)propanoic acid hydrochloride | 625120-81-2 | 伊班膦酸钠中间体 | |
20 | IBAN-1 | 伊班膦酸钠 | Ibandronate Sodium | 138926-19-9 | API |